GDC-0980 (Apitolisib)
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Technical Data
Description
GDC-0980 (Apitolisib) is a potent dual PI3 kinase/mTOR inhibitor. GDC-0980 inhibits both PI3K kinase and mTOR kinase, which may result in tumor cell apoptosis and growth inhibition of cancer cells overexpressing PI3K/mTOR.