GDC-0980 (Apitolisib)

SKU: C-1149-5mg

Quantity (mg):

5 mg

Product Options

Quantity

$103.99

Catalog#: C-1149

Targets: PI3K

Synonym: GDC0980; GDC-0980; GDC 0980; RG7422; RG-7422; RG 7422; GNE 390; GNE-390; GNE390; Apitolisib

Chemical Name/IUPAC:(S)-1-(4-((2-(2-aminopyrimidin-5-yl)-7-methyl-4-morpholinothieno[3,2-d]pyrimidin-6-yl)methyl)piperazin-1-yl)-2-hydroxypropan-1-one

Technical Data

Product Name: GDC-0980 (Apitolisib)

Chemical Formula: C23H30N8O3S

Molecular Weight: 498.6

CAS#: 1032754-93-0

Appearance: Solid powder

Purity: > 99% by HPLC

Solubility: Soluble in DMSO

Storage: Room temperature for months, or -20ºC for 3 years

Description
GDC-0980 (Apitolisib) is a potent dual PI3 kinase/mTOR inhibitor. GDC-0980 inhibits both PI3K kinase and mTOR kinase, which may result in tumor cell apoptosis and growth inhibition of cancer cells overexpressing PI3K/mTOR.

GDC-0980 (Apitolisib)

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