Enzalutamide (MDV-3100)

SKU: C-1376-5mg

Quantity (mg):

250 mg

Product Options

Quantity

$227.00

Catalog#: C-1376

Quantity: 5mg

Targets: Androgen Receptor (AR)

Synonym: MDV3100; MDV 3100; MDV-3100; Enzalutamide

Chemical Name/IUPAC:4-(3-(4-cyano-3-(trifluoromethyl)phenyl)-5,5-dimethyl-4-oxo-2-thioxoimidazolidin-1-yl)-2-fluoro-N-methylbenzamide

SMILES Code: O=C(NC)C1=CC=C(N(C(N2C3=CC=C(C#N)C(C(F)(F)F)=C3)=S)C(C)(C)C2=O)C=C1F

Technical Data

Product Name: Enzalutamide (MDV-3100)

Chemical Formula: C21H16F4N4O2S

Molecular Weight: 464.43

CAS#: 915087-33-1

Purity: > 99% by HPLC

Solubility: Soluble in DMSO

Storage: Room temperature for months, or -20ºC for 3 years

Description
Enzalutamide (MDV-3100) is an orally bioavailable, organic, non-steroidal small molecule targeting the androgen receptor (AR) with potential antineoplastic activity. Through a mechanism that is reported to be different from other approved AR antagonists, selective androgen receptor modulator MDV3100 inhibits the activity of prostate cancer cell ARs, which may result in a reduction in prostate cancer cell proliferation and, correspondingly, a reduction in the serum prostate specific antigen (PSA) level.

Enzalutamide (MDV-3100)

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